2019 Original Papers / 2019 原著論文
- Yamada, D.; Yanagisawa, S.; Yoshizawa, K.; Yanagita, S.; Oka, J.; Nagase, H.; Saitoh, A.
“Selective agonists of the δ-opioid receptor, KNT-127 and SNC80, act differentially on extinction learning of contextual fear memory in mice”
Neuropharmacology 2019, 160, 107792. (web) - Saitoh, T.; Seki, K.; Nakajima, R.; Yamamoto, N.; Kutsumura, N.; Nagumo, Y.; Irukayama-Tomobe, Y.; Ogawa, Y.; Ishikawa, Y.; Tanimura, R.; Yanagisawa, M.; Nagase, H.
“Essential structure of orexin 1 receptor antagonist YNT-707, Part IV: The role of D-ring in 4,5-epoxymorphinan on the orexin 1 receptor antagonistic activity”
Bioorg. Med. Chem. Lett. 2019, 29, 2655-2658. (web) - Kutsumura, N.; Inagaki, M.; Kiriseko, A.; Saito, T.
“Total Synthesis of 3-epi-Juruenolide C”
Chem. Pharm. Bull. 2019, 67, 594-598. (web)
selected as a Highlighted paper selected by Editor-in-Chief.
selected as a Featured Article.
- Yamamoto, N.; Ohrui, S.; Okada, T.; Saitoh, T.; Kutsumura, N.; Nagumo, Y.; Irukayama-Tomobe, Y.; Ogawa, Y.; Ishikawa, Y.; Watanabe, Y.; Hayakawa, D.; Gouda, H.; Yanagisawa, M.; Nagase, H.
“Essential structure of orexin 1 receptor antagonist YNT-707, Part III: Role of the 14-hydroxy and the 3-methoxy groups in antagonistic activity toward the orexin 1 receptor in YNT-707 derivatives lacking the 4,5-epoxy ring”
Bioorg. Med. Chem. 2019, 27, 1747-1758. (web) (Invited Paper) - Yata, M.; Kutsumura, N.; Nagumo, Y.; Yamamoto, N.; Saitoh, T.; Ishikawa, Y.; Irukayama-Tomobe, Y.; Yanagisawa, M.; Nagase, H.
“A Novel Rearrangement Reaction of Morphinan to Arylmorphan Skeletons and the Pharmacologies of Arylmorphan Derivatives”
Heterocycles 2019, 99, 134-144. (web) (Invited Paper) - Hirayama, S.; Obayashi, K.; Wada, N.; Ohyama, K.; Fuku, S.; Koyano, K.; Karaki, F.; Itoh, K.; Nagase, H.; Fujii, H.
“The Practical Synthesis of Dissymmetrical 1,3,5-Trioxazatriquinane Derivatives Comprised of Three Distinct Carbonyl Compounds”
Heterocycles 2019, 99, 1003-1019. (web) (Invited Paper)
- Kutsumura, N.; Numata, K.; Mosaki, S.; Saito, T.
“Total Synthesis of Haplacutines B and C”
Heterocycles 2019, 99, 614-624. (web) (Invited Paper)
- Korkutata, M.; Saitoh, T.; Cherasse, Y.; Ioka, S.; Duo, F.; Qin, R.; Murakoshi, N.; Fujii, S.; Zhou, X.; Sugiyama, F.; Chen, J.-F.; Kumagai, H.; Nagase, H.; Lazarus, M.
“Enhancing endogenous adenosine A2A receptor signaling induces slow-wave sleep without affecting body temperature and cardiovascular function”
Neuropharmacol. 2019, 144, 122-132. (web) - Sugiyama, A.; Yamada, M.; Furuie, H.; Gotoh, L.; Saitoh, A.; Nagase, H.; Oka, J.; Yamada, M.
“Systemic administration of a delta opioid receptor agonist, KNT-127, facilitates extinction learning of fear memory in rats”
J. Pharmacol. Sci. 2019, 139, 174-179. (web) - Zhang, Y.; Sugai, T.; Yamamoto, T.; Yamamoto, N.; Kutsumura, N.; Nishiyama, S.; Einaga, Y.; Saitoh, T.; Nagase, H.
“Oxidative Cleavage of the Acyl-Carbon Bond in Phenylacetone with Electrogenerated Superoxide Anions”
ChemElectroChem 2019, 6, 4194-4198. (web) (Invited Paper)